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Product Name: Cetirizine
Generic Name: Cetirizine
Common Brands: Zyrtec
Pharmaceutical Categories: Anti-Allergic, Asthma
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Cetirizine (trade names include Zyrtec, Adezio, Alatrol, Alerid, Alerlisin, All Day Allergy, Allercet, Allergy Relief, Allerkid, Alzytec, Apo-Cetirizine, Benadryl Allergy, Benadryl One A Day, Cerzin, Cetallerg, Cetcip, Cetgel, Cetiristad, Cetrizet, Cetzine, Drill Allergie, Formistin, Glotrizine, Hayfever and Allergy Relief, Histacet, Histazine, Humex Allergie, Incidal-OD, Lerzin, Letizen, Okacet, Piriteze Allergy, Quzyttir, Reactine, Reactine Allergy, Rhizin, Sinutab Sinus Allergy, Talerc, Tiriz, Virlix, Zanlan, Zyllergy, Zyncet, Zyrlex, Zyrtec Allergy, Zyrtec Children's Allergy, ZyrtecSet) is a second-generation non-drowsy antihistamine (anti-allergic) medicine from piperazine derivatives pharmacological group. This medication is used for the treatment or prevention symptoms of allergies, dermatitis, acute and chronic urticaria (hives), eustachian tube dysfunction. It also indicated to relief symptoms associated with seasonal and perennial allergic rhinitis, hay fever due to allergens such as ragweed, grass and tree pollens, dust mites, animal dander and molds. The therapy of symptoms is effective for sneezing, itchy, runny nose; itchy, red, watery eyes in adults and children. Cetirizine works by reducing the natural chemical histamine in the body. Zyrtec provides allergy relief up to 24 hours.
Related medications:
Azelastine (Astelin)
Bilastine (Ilaxten)
Buclizine (Longifene)
Budesonide (Entocort, Rhinocort)
Chlorcyclizine (Ahist)
Cyclizine (Valoid)
Cyproheptadine (Periactin)
Danazol (Danocrine)
Desloratadine (Clarinex)
Dexamethasone (Decadron, Dexone)
Fexofenadine (Allegra)
Fluticasone (Flonase)
Hydrocortisone (Cortef, Locoid)
Hydroxyzine (Atarax)
Ketotifen (Zaditor)
Levocetirizine (Xyzal)
Loratadine (Claritin)
Meclizine (Antivert)
Mometasone (Elocon, Nasonex)
Montelukast (Singulair)
Olopatadine (Patanol)
Oxatomide (Tinset)
Promethazine (Phenergan)
Triamcinolone (Aristocort)
Pharmaceutical and medical classifications:
Anti allergic medications
Antiallergic agents
Antihistamine drugs
H1-antihistaminics
Histamine H1-receptor antagonists
One a day allergy tablets
Peripheral H1-blockers
Piperazines
Second-generation antihistamines
The Anatomical Therapeutic Chemical (ATC) classification system (developed by the World Health Organization):
R - Respiratory system
R06 - Antihistamines for systemic use
R06A - Antihistamines for systemic use
R06AE - Piperazine derivatives
R06AE07 - Cetirizine
S - Sensory organs
S01 - Ophthalmologicals
S01G - Decongestants and antiallergics
S01GX - Other antiallergics
S01GX12 - Cetirizine
Medical conditions for cetirizine in the International Statistical Classification of Diseases and Related Health Problems (ICD):
Conjunctivitis - H10
Chronic conjunctivitis - H10.4
Other disorders of eye and adnexa - H57
Other specified disorders of eye and adnexa - H57.8
Other and unspecified disorders of Eustachian tube - H69
Acute bronchiolitis - J21
Vasomotor and allergic rhinitis - J30
Allergic rhinitis due to pollen - J30.1
Other allergic rhinitis - J30.8
Allergic rhinitis due to animal (cat) (dog) hair and dander - J30.81
Other allergic rhinitis - J30.89
Allergic rhinitis, unspecified - J30.9
Atopic dermatitis - L20
Allergic contact dermatitis - L23
Irritant contact dermatitis - L24
Lichen simplex chronicus and prurigo - L28
Pruritus - L29
Other dermatitis - L30
Urticaria - L50
Other urticaria - L50.8
Urticaria, unspecified - L50.9
Abnormalities of breathing - R06
Sneezing - R06.7
Other symptoms and signs involving the circulatory and respiratory system - R09
Other specified symptoms and signs involving the circulatory and respiratory systems - R09.8
Nasal congestion - R09.81
Rash and other nonspecific skin eruption - R21
Adverse effects, not elsewhere classified - T78
Pregnancy category:
B2 - Australia
B - United States (No evidence of risk in humans)
Forms of active pharmaceutical ingredients (APIs):
Cetirizine Base
Cetirizine Dihydrochloride
Cetirizine Hydrochloride
Chemical, international, and other names of this drug:
Acetic acid, [2-[4-[(4-chlorophenyl)phenylmetyl]-1-piperazinyl]etoxy]-
Cetirizin
Cetirizin Dihydrochlorid
Cetirizin Hydrochlorid
Cetirizina
Cetirizina Diclorhidrato
Cetirizin-Dihidroklorid
Cetirizindihydrochlorid
Cetirizine 2HCl
Cetirizine Dichlorhydrate
Cetirizine HCl
Cetirizinedihydrochloride
Cetirizini Dihydrochloridum
Cetirizinum
Cetrizine
Cetyryzyna
Clorhidrato de Cetirizina
Cloridrato de Cetirizina
Diclorhidrato de Cetirizina
Setiritsiini
Setiritsiinidihydrokloridi
Setirizin
Most known trade names (brands and generics) worldwide:
Aceterin - Sandoz, Hexal
Acidrine - Novamed Laboratorio
Actifed Allergie - Pfizer, Johnson & Johnson, Ortho McNeil Pharmaceuticals
Acuzyrt - Cipla
Adezio - Xepa-Soul Pattinson, Apex Pharma Marketing, Four Star, Grafton Pharmasia, KTZ, Tack Fung Medical Supplies
Agelmin - Kleva, CDL Pharmaceutical, Drug Houses of Australia
Alairgix - Cooperation Pharmaceutique Francaise
Alatrol - Square Pharmaceuticals, Medispec
Alercina - Cinfa Laboratorios
Alerid - Cipla, Chiesi, CZ Pharma, Pharmatec Pakistan, S & D Pharma CZ, Terapia, UCB Pharma
Alerlisin - Menarini
Alertop - Chile Laboratorios
Alerzina - Lek-Am Przedsiebiorstwo Farmaceutyczne
All Day Allergy - Major Pharmaceuticals
Allecet - Cipla
Allercet - Micro Labs, Brown & Burk Pharmaceuticals, Cosma Medical, Zizawa Healthcare
Allergietabletten - Healthypharm
Allergy Relief - Apotex
Allergy Care - Trima Pharmaceuticals
Allerkid - Pediatrica, United Laboratories
Aller-Tec - Costco Wholesale Company
Allertec - Polfa Warszawa, Pharmacare, Ziwell Medical
Alnok - Sandoz, DuraScan Medical Products
Alzene - Alphapharm
Alzytec - Samchully Pharm, Zyfas Medical
Amertil Bio - Biofarm
Apo-Cetirizine - Apotex
Avil NU - Sanofi
Baydal - Bayer
Benaday - Pfizer, Ortho McNeil Pharmaceuticals
Benadryl Allergy - Pfizer, Ortho McNeil Pharmaceuticals
Benadryl Allergy Children's - Pfizer, Ortho McNeil Pharmaceuticals
Benadryl One A Day - Pfizer, Johnson & Johnson
Celerg - A.C. Helcor
Cerini - Sanbe Farma
Cerzin - Mepha
CetAlergin - Valeant Pharmaceuticals, PharmaSwiss
Cetallerg - Sandoz, Ecosol
Cetcip - Cipla
Cetgel - Universal Medicare
Cetigran - Axxon
Cetinal - Kalbe Farma
Cetiristad - Stada
Cetirivax - Vivax Pharmaceuticals
Cetiriz - Alkem Laboratories, Pyrex Trading, Zifam Pinnacle
Cetirizin - 1 A Pharma, AbZ-Pharma, Actavis, Basics, Bluefish Pharmaceuticals, BMM Pharma, CT-Arzneimittel, Genericon Pharma, Generics UK, Heumann Pharma, Hexal, Mylan, Ratiopharm, Sandoz, Stada, Zentiva
Cetirizina - Actavis, Alter Laboratorios, Apotex, Calox International, Cinfa Laboratorios, DOC Generici, Generis Farmaceutica, Genfar Laboratorios, Kern Pharma, La Sante Laboratorios, Medley Industria Farmaceutica, Mylan, Normon Laboratorios, Ranbaxy, Ratiopharm, Sandoz, Teva, Zentiva
Cetirizindihydrochlorid - Stada
Cetirizine - Actavis, Arrow Generiques, Biogaran, Cipla, EG Labo, Generics UK, Mylan, Ratiopharm, Sandoz, Stada, Teva, UCB Pharma
Cetirizine Allergy - Apotex, Dr. Reddy's Laboratories, Sun Pharmaceutical Industries, Wockhardt
Cetirizine Conseil - Arrow Generiques, Ratiopharm, Teva
Cetirizinedihydrochloride - Ratiopharm
Cetirizinum - Synoptis Pharma
CetiSandoz - Sandoz
Cetril - Brussels Laboratories
Cetriler - Roux-Ocefa Laboratorios
Cetrizet - Sun Pharmaceutical Industries
Cetryn - Tripharma Ilac
Cettec - Medicpharma
Cetzine - Dr. Reddy's Laboratories
Cezil - Sanofi, Ampharco
Children's All Day Allergy - Major Pharmaceuticals
Children's Zyrtec Allergy - Pfizer, Johnson & Johnson, Ortho McNeil Pharmaceuticals
Coolips - Mintlab
Curtec - Bottu Laboratoires
CZ 3 - Lupin
Drill Allergie - Pierre Fabre
Extra Strength Allergy Relief - PendoPharm, Pharmascience
Falergi - Fahrenheit, Pratapa Nirmala
Finallerg - Pharma International Company
Findaler - Medipharm Productos Farmaceuticos
Formistin - Istituto Luso Farmaco d'Italia
Glotrizine - Global Pharma
Hayfever and Allergy Relief - Boots, Lloyds Pharmacy
Hayfever Relief - Peach Ethical
Hicet - Micro Labs
Hisaler - Bago Laboratorios
Histacet - Medreich, DKSH
Histacet - Merril Pharma
Histazine - Trima Pharmaceuticals, Amriya Pharmaceutical Industries, Gaily Pharmaceutical
Histrine - Ferron
Hitrizin - Deva Holding Ilac Grubu
Humex Allergie - Urgo Laboratoires
Incid-L - Bayer, Zydus Pharmaceuticals
Incidal-OD - Bayer
Intazin - Intas Pharmaceuticals
Intrizin - Interbat
Lerzin - Ifars Pharmaceutical Laboratories
Letizen - KRKA
Miseda - Atlantis
Okacet - Cipla
Optiser - Apotecarium
Parlazin - Egis, Mekim
Piriteze Allergy - GlaxoSmithKline
PMS-Cetirizine - Pharmascience
Quzyttir - TerSera Therapeutics
RatioAllerg - Ratiopharm
Reactine - Pfizer, Johnson & Johnson, Ortho McNeil Pharmaceuticals, UCB Pharma
Reactine Allergy - Pfizer, Ortho McNeil Pharmaceuticals
Revicet - Sager Pharma
Rhinodina - Alexxia Pharma, Roddome Pharmaceutical
Rhizin - Zydus Cadila Healthcare, Cibex, Zyfas Medical
Rigix - UCB Pharma, AGP
Rigotax - Prater Laboratorio, Qualipharm
Rinalgit - ABC Farmaceutici
Rinazina - Pliva, Labiana Pharmaceuticals
Ryvel - Novell Pharmaceutical Laboratories, CNW Hong Kong, Hong Tai Hong
Salvalerg - GlaxoSmithKline
Sandoz Cetirizine - Sandoz
Sinutab Sinus Allergy - Johnson & Johnson
Stopaler - LKM Laboratorio
Tabcin Alergi - Bayer
Talerc - Boehringer Ingelheim
Talerdin - Gutis Productos
Talzic - Elmor Laboratorios
Tiriz - Lapi Laboratories
Triofan Allergie - Vifor Pharma
Vialerg - Orifarm
Virlix - Sanofi, Farchim, GlaxoSmithKline, Grunenthal, Lacer, Mediolanum Farmaceutici, UCB Pharma, Vedim Pharma, Zuellig Pharma
Zadryl - Polymedic Trading Enterprise
Zanlan - Novartis, Salutas Pharma, Sandoz
Zetalerg - UCI-Farma Industria Farmaceutica
Zetop - Actavis, Alliance Pharmaceuticals, Zydus Cadila Healthcare
Zirtec - UCB Pharma
Zirtek - UCB Pharma, Hansel Pharmacueutical, United Drug
Zyllergy - Dexxon
Zyncet - Torrent Pharmaceuticals, Unichem Laboratories
Zyrlex - UCB Pharma, Macure Pharma
Zyrtec - Pfizer, Adon Pharmaceuticals, Aesica Pharmaceuticals, AGP, Armstrong Laboratorios de Mexico, BCN Farma, Beragena Arzneimittel, Bryant Ranch Prepack, Dexxon, Dr. Fisher Farma, Dr. Reddy's Laboratories, Duncan Pharmaceuticals, Ecosse Pharmaceuticals, Emra-Med Arzneimittel, Firma Chun Cheong, GlaxoSmithKline, Johnson & Johnson, Kenvue Brands, Kohlpharma, NeoFarma Pharmaceuticals, Olic Thailand, Opti-Arznei, Ortho McNeil Pharmaceuticals, Pharmabroker Sales, Pliva, Rontag Laboratorios, UCB Pharma, Zuellig Pharma
Zyrtec Allergy - Pfizer, Johnson & Johnson, Ortho McNeil Pharmaceuticals
Zyrtec Children's Allergy - Pfizer, Johnson & Johnson, Ortho McNeil Pharmaceuticals
Zyrtec Hives Relief - Pfizer, Johnson & Johnson, Ortho McNeil Pharmaceuticals
Zyrtec Infantil - Pfizer
ZyrtecSet - Pfizer, Pierre Fabre
Other medicines used in combinations with cetirizine:
Acetaminophen
Albuterol
Ambroxol
Ammonium Chloride
Bromhexine
Caffeine
Chlorpheniramine
Dextromethorphan
Diethylcarbamazine
Guaifenesin
Menthol
Montelukast
Nimesulide
Phenylephrine
Phenylpropanolamine
Pseudoephedrine
Zinc Gluconate
References and external sources:
Cetirizine main article on Wikipedia: https://en.wikipedia.org/wiki/Cetirizine
Cetirizine compound on PubChem: https://pubchem.ncbi.nlm.nih.gov/compound/Cetirizine
Cetirizine Hydrochloride on PubChem: https://pubchem.ncbi.nlm.nih.gov/compound/Cetirizine-Hydrochloride
Cetirizine medicine on DrugBank: https://go.drugbank.com/drugs/DB00341
Cetirizine FAQ on MedlinePlus (revised 10/15/2023): https://medlineplus.gov/druginfo/meds/a623043.html
Cetirizine Injection on MedlinePlus (revised 12/15/2022): https://medlineplus.gov/druginfo/meds/a698026.html
Zyrtec (Cetirizine Hydrochloride) film-coated tablets drug label on DailyMed (revised April 28, 2015): https://dailymed.nlm.nih.gov/dailymed/drugInfo...
Zyrtec (Cetirizine Hydrochloride) capsules drug label on DailyMed (revised November 8, 2024): https://dailymed.nlm.nih.gov/dailymed/drugInfo...
Amneal Cetirizine Hydrochloride tablets drug label on DailyMed (revised July 31, 2024): https://dailymed.nlm.nih.gov/dailymed/drugInfo...
Zyrtec (Cetirizine Hydrochloride) tablets and syrup for oral use official prescribing information from the U.S. FDA (revised 01/2002): https://www.accessdata.fda.gov/drugsatfda_docs/label/...
Zyrtec (Cetirizine Hydrochloride) official website powered by Kenvue Brands LLC: https://www.zyrtec.com/
Allergy Relief (Cetirizine Hydrochloride tablets 5 mg) and Extra Strength Allergy Relief (Cetirizine Hydrochloride tablets 10 mg) product monograph and consumer information from The Drug and Health Product Register (revised August 17, 2018): https://pdf.hres.ca/dpd_pm/00046970.PDF
Zyrtec (Cetirizine Hydrochloride) tablets, oral liquid, oral drops product information from Medicines.org.au (revised May 2019): https://apps.medicines.org.au/files/pcpzyrtc.pdf
Zirtek Allergy (Cetirizine Hydrochloride) 10 mg film-coated tablets package information leaflet for uses from Medicines.org.uk (revised 09/2023): https://www.medicines.org.uk/emc/files/pil.6751.pdf
Revised: March 2025
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